Middendorp, Simon

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Middendorp, Simon; Maldifassi, Maria Constanza; Baur, Roland; Sigel, Erwin (2015). Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site. Neuropharmacology, 95, pp. 459-467. Elsevier 10.1016/j.neuropharm.2015.04.027

Middendorp, Simon; Hurni, Evelyn; Schönberger, Matthias; Stein, Marco; Pangerl, Michael; Trauner, Dirk; Sigel, Erwin (2014). Relative positioning of classical benzodiazepines to the γ2-subunit of GABAA receptors. ACS Chemical Biology, 9(8), pp. 1846-1853. American Chemical Society 10.1021/cb500186a

Middendorp, Simon; Puthenkalam, Roshan; Baur, Roland; Ernst, Margot; Sigel, Erwin (2014). Accelerated discovery of novel benzodiazepine ligands by experiment-guided virtual screening. ACS Chemical Biology, 9(8), pp. 1854-1859. American Chemical Society 10.1021/cb5001873

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