ChemMedChem

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Number of items: 21.

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Kopp, Sascha; Baur, Roland; Sigel, Erwin; Möhler, Hanns; Altmann, Karl-Heinz (2010). Highly potent modulation of GABA(A) receptors by valerenic acid derivatives. ChemMedChem, 5(5), pp. 678-81. Weinheim: Wiley-VCH 10.1002/cmdc.201000062

Erdélyi, Máté; Navarro-Vázquez, Armando; Pfeiffer, Bernhard; Kuzniewski, Christian N; Felser, Andrea; Widmer, Toni; Gertsch, Jürg; Pera, Benet; Díaz, José Fernando; Altmann, Karl-Heinz; Carlomagno, Teresa (2010). The binding mode of side chain- and C3-modified epothilones to tubulin. ChemMedChem, 5(6), pp. 911-920. Weinheim: Wiley-VCH 10.1002/cmdc.201000050

van Deursen, Ruud; Reymond, Jean-Louis (2007). Chemical Space Travel. ChemMedChem, 2(5), pp. 636-640. Weinheim: Wiley-VCH 10.1002/cmdc.200700021

Nguyen, Kong Thong; Syed, Salahuddin; Urwyler, Stephan; Bertrand, Sonia; Bertrand, Daniel; Reymond, Jean-Louis (2008). Discovery of NMDA Glycine Site Inhibitors from the Chemical Universe Database GDB. ChemMedChem, 3(10), pp. 1520-1524. Weinheim: Wiley-VCH 10.1002/cmdc.200800198

Nguyen, Kong Thong; Blum, Lorenz C.; van Deursen, Ruud; Reymond, Jean-Louis (2008). Classification of Organic Molecules by Molecular Quantum Numbers (Communication). ChemMedChem, 4(11), pp. 1803-1805. Weinheim: Wiley-VCH 10.1002/cmdc.200900317

Kolomiets, Elena; Swiderska, Magdalena A.; Kadam, Rameshwar U.; Johansson, Emma M.V.; Jaeger, Karl-Erich; Darbre, Tamis; Reymond, Jean-Louis (2009). Glycopeptide dendrimers with high affinity for the fucose binding lectin PA-IIL from Pseudomonas aeruginosa. ChemMedChem, 4(4), pp. 562-569. Weinheim: Wiley-VCH 10.1002/cmdc.200800380

Berger, Isabella; Nazarov, Alexey A.; Hartinger, Christian G.; Grössl, Michael; Valiahdi, Seied-M.; Jakupec, Michael A.; Keppler, Bernhard K. (2007). A glucose derivative as natural alternative to the cyclohexane-1,2-diamine ligand in the anticancer drug oxaliplatin? ChemMedChem, 2(4), pp. 505-514. Wiley-VCH 10.1002/cmdc.200600279

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Pujol-Giménez, Jonai; Poirier, Marion; Bühlmann, Sven; Schuppisser, Céline; Bhardwaj, Rajesh; Awale, Mahendra; Visini, Ricardo; Javor, Sacha; Hediger, Matthias; Reymond, Jean-Louis (2021). Inhibitors of Human Divalent Metal Transporters DMT1 (SLC11A2) and ZIP8 (SLC39A8) from a GDB-17 Fragment Library. ChemMedChem, 16(21), pp. 3306-3314. Wiley-VCH 10.1002/cmdc.202100467

Zakharova, Elena; Orsi, Markus; Capecchi, Alice; Reymond, Jean-Louis (2022). Machine Learning Guided Discovery of Non-Hemolytic Membrane Disruptive Anti-Cancer Peptides. ChemMedChem, 17(17), e202200291. Wiley-VCH 10.1002/cmdc.202200291

Graff, Julien; Müller, Jennifer; Sadurní, Anna; Rubin, Matthias; Cuissa, Inês André Canivete; Keller, Claudia; Hartmann, Marco; Singer, Simon; Gertsch, Jürg; Altmann, Karl-Heinz (2022). The Evaluation of L-Tryptophan Derivatives as Inhibitors of the LType Amino Acid Transporter LAT1 (SLC7A5). ChemMedChem, 17(17), e202200308. Wiley-VCH 10.1002/cmdc.202200308

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Fuhrer, Cyril; Grüter, Eric; Ruetz, Stephan; Häner, Robert (2007). Cis-Stilbene Derived Furopyranones Show Potent Antiproliferative Activity by Inducing G2/M Arrest. ChemMedChem, 2(4), pp. 441-444. Weinheim: Wiley-VCH 10.1002/cmdc.200600284

Koceva-Chyła, Aneta; Matczak, Karolina; Hikisz, Msc. Paweł; Durka, Msc. Kamil; Kochel, Msc. Krzysztof; Süss-Fink, Georg; Furrer, Julien; Kowalski, Konrad (2016). Insights into the in vitro Anticancer Effects of Diruthenium-1. ChemMedChem, 11(19), pp. 2171-2187. Wiley-VCH 10.1002/cmdc.201600315

Probst, Daniel; Heitz, Marc; Poirier, Marion; Gan, Bee Ha; Delalande, Clémence Marie Sandrine; Reymond, Jean-Louis (2017). Frontiers in Medicinal Chemistry 2017 in Bern, Switzerland. ChemMedChem, 12(19), pp. 1645-1651. Wiley-VCH 10.1002/cmdc.201700306

Cubo, Leticia; Grössl, Michael; Dyson, Paul J.; Quiroga, Adoración G.; Navarro-Ranninger, Carmen; Casini, Angela (2010). Proteins as Possible Targets for Cytotoxic trans-Platinum(II) Complexes with Aliphatic Amine Ligands: Further Exceptions to the DNA Paradigm. ChemMedChem, 5(8), pp. 1335-1343. Wiley-VCH 10.1002/cmdc.201000104

Harmse, Rozanne; Wong, Ho Ning; Smit, Frans J; Müller, Joachim; Hemphill, Andrew; N'Da, David D; Haynes, Richard K (2017). Activities of 11-Azaartemisinin and N-Sulfonyl Derivatives against Neospora caninum and Comparative Cytotoxicities. ChemMedChem, 12(24), pp. 2094-2098. Wiley-VCH 10.1002/cmdc.201700600

Lin, Arkadii; Horvath, Dragos; Afonina, Valentina; Marcou, Gilles; Reymond, Jean-Louis; Varnek, Alexandre (2018). Mapping of the Available Chemical Space versus the Chemical Universe of Lead-Like Compounds. ChemMedChem, 13(6), pp. 540-554. Wiley-VCH 10.1002/cmdc.201700561

Poirier, Marion; Awale, Mahendra; Rölli, Matthias A.; Giuffredi, Guy T.; Ruddigkeit, Lars; Evensen, Lasse; Stooss, Amandine; Calarco, Serafina; Lorens, James B.; Charles, Roch-Philippe; Reymond, Jean-Louis (2018). Identifying Lysophosphatidic Acid Acyltransferase β (LPAAT-β) as the Target of a Nanomolar Angiogenesis Inhibitor from a Phenotypic Screen Using the Polypharmacology Browser PPB2. ChemMedChem, 14(2), pp. 224-236. Wiley-VCH 10.1002/cmdc.201800554

Petruk, Ganna; Monti, Daria Maria; Ferraro, Giarita; Pica, Andrea; D'Elia, Luigi; Pane, Francesca; Amoresano, Angela; Furrer, Julien; Kowalski, Konrad; Merlino, Antonello (2019). Encapsulation of the dinuclear trithiolato-bridged arene ruthenium complex diruthenium-1 in an apoferritin nanocage: structure and cytotoxicity. ChemMedChem, 14(5), pp. 594-602. Wiley-VCH 10.1002/cmdc.201800805

Bartholomäus, Ruben; Nicolussi, Simon; Baumann, Alice; Rau, Mark; Simão, Ana Catarina; Gertsch, Jürg; Altmann, Karl-Heinz (2019). Total Synthesis of the Endocannabinoid Uptake Inhibitor Guineensine and SAR Studies. ChemMedChem, 14(17), pp. 1590-1596. Wiley-VCH 10.1002/cmdc.201900390

Mäder, Patrick; Bartholomäus, Ruben; Nicolussi, Simon; Baumann, Alice; Weis, Melanie; Chicca, Andrea; Rau, Mark; Simão, Ana Catarina; Gertsch, Jürg; Altmann, Karl-Heinz (2021). Synthesis and Biological Evaluation of Endocannabinoid Uptake Inhibitors Derived from WOBE437. ChemMedChem, 16(1), pp. 145-154. Wiley-VCH 10.1002/cmdc.202000153

Schuppisser, Céline; Mulliri, Kleni (2024). Drug Discovery Summit: 14 th Swiss Course on Medicinal Chemistry. ChemMedChem, 19(4), e202300579. Wiley 10.1002/cmdc.202300579

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