Gertsch, Jürg

No

Bátora, Dániel; Fischer, Jérôme P.; Kaderli, Reto M.; Varga, Maté; Lochner, Martin; Gertsch, Jürg (25 February 2024). Silicon-rhodamine functionalized evocalcet probes (EvoSiR) potently and selectively label calcium sensing receptors (CaSR) in vitro, in vivo and ex vivo (bioRxiv). Cold Spring Harbor Laboratory 10.1101/2024.02.22.581561

Gertsch, Jürg (2021). Travelogues from the Rainforest: Notes on Prof. Otto Sticher's 85th birthday. Planta medica, 87(14), pp. 1123-1127. Thieme 10.1055/a-1508-0613

Gertsch, Jürg (2018). Analytical and Pharmacological Challenges in Cannabis Research. Planta medica, 84(4), p. 213. Thieme 10.1055/s-0044-101051

Feyen, Fabian; Cachoux, Frédéric; Gertsch, Jürg; Wartmann, Markus; Altmann, Karl-Heinz (2008). Epothilones as lead structures for the synthesis-based discovery of new chemotypes for microtubule stabilization. Accounts of chemical research, 41(1), pp. 21-31. Easton, Pa.: American Chemical Society 10.1021/ar700157x

Yes

Gertsch, Jürg; Chicca, Andrea (2024). CNS Drug Discovery in Academia: Where Basic Research Meets Innovation. ChemBioChem, 25(19), e202400397. Wiley 10.1002/cbic.202400397

Kroll, Sara L; Meier, Philip; Mayo, Leah M; Gertsch, Jürg; Quednow, Boris B (2024). Endocannabinoids and related lipids linked to social exclusion in individuals with chronic non-medical prescription opioid use. Neuropsychopharmacology, 49(10), pp. 1630-1639. Springer Nature 10.1038/s41386-024-01881-8

Hirschi, Stephan; Lemmin, Thomas; Ayoub, Nooraldeen; Kalbermatter, David; Pellegata, Daniele; Ucurum, Zöhre; Gertsch, Jürg; Fotiadis, Dimitrios (2024). Structural insights into the mechanism and dynamics of proteorhodopsin biogenesis and retinal scavenging. Nature Communications, 15(1), p. 6950. Springer Nature 10.1038/s41467-024-50960-3

Chicca, Andrea; Bátora, Daniel; Ullmer, Christoph; Caruso, Antonello; Grüner, Sabine; Fingerle, Jürgen; Hartung, Thomas; Degen, Roland; Müller, Matthias; Grether, Uwe; Pacher, Pal; Gertsch, Jürg (2024). A Highly Potent, Orally Bioavailable Pyrazole-Derived Cannabinoid CB2 Receptor- Selective Full Agonist for In Vivo Studies. ACS pharmacology & translational science, 7(8), pp. 2424-2438. ACS Publications 10.1021/acsptsci.4c00269

Bátora, Dániel; Dienes-Nagy, Ágnes; Zeng, Liming; Gerber, Christian E.; Fischer, Jérôme P.; Lochner, Martin; Gertsch, Jürg (2024). Hypersensitive quantification of major astringency markers in food and wine by substoichiometric quenching of silicon-rhodamine conjugates. Food Chemistry: X, 23, p. 101592. Elsevier 10.1016/j.fochx.2024.101592

Tomašević, Nataša; Emser, Fabiola Susanna; Muratspahić, Edin; Gattringer, Jasmin; Hasinger, Simon; Hellinger, Roland; Keov, Peter; Felkl, Manuel; Gertsch, Jürg; Becker, Christian F W; Gruber, Christian W (2024). Discovery and development of macrocyclic peptide modulators of the cannabinoid 2 receptor. The journal of biological chemistry, 300(6), p. 107330. American Society for Biochemistry and Molecular Biology 10.1016/j.jbc.2024.107330

Chicca, Andrea; Batora, Daniel; Ullmer, Christoph; Caruso, Antonello; Fingerle, Jürgen; Hartung, Thomas; Degen, Roland; Müller, Matthias; Grether, Uwe; Pacher, Pal; Gertsch, Jürg (29 April 2024). A highly potent, orally bioavailable pyrazole-derived cannabinoid CB2 receptor-selective full agonist for in vivo studies. (bioRxiv). Cold Spring Harbor Laboratory 10.1101/2024.04.26.591311

Bátora, Daniel; Fischer, Jérôme P.; Kaderli, Reto M.; Varga, Máté; Lochner, Martin; Gertsch, Jürg (2024). Silicon-Rhodamine Functionalized Evocalcet Probes Potently and Selectively Label Calcium Sensing Receptors In Vitro, In Vivo, and Ex Vivo. ACS pharmacology & translational science, 7(5), pp. 1557-1570. ACS Publications 10.1021/acsptsci.4c00096

Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; ... (2024). Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors. European journal of medicinal chemistry, 263(115916), p. 115916. Elsevier 10.1016/j.ejmech.2023.115916

Alexander, Stephen P H; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair A; Peters, John A; Veale, Emma L; Armstrong, Jane F; Faccenda, Elena; Harding, Simon D; Davies, Jamie A; Annett, Stephanie; Boison, Detlev; Burns, Kathryn Elisa; Dessauer, Carmen; Gertsch, Jurg; Helsby, Nuala Ann; Izzo, Angelo A; Ostrom, Rennolds; Papapetropoulos, Andreas; Pyne, Nigel J; ... (2023). The Concise Guide to PHARMACOLOGY 2023/24: Enzymes. British journal of pharmacology, 180 Suppl 2, S289-S373. Wiley-Blackwell 10.1111/bph.16181

Maccarrone, Mauro; Di Marzo, Vincenzo; Gertsch, Juerg; Grether, Uwe; Howlett, Allyn C; Hua, Tian; Makriyannis, Alexandros; Piomelli, Daniele; Ueda, Natsuo; van der Stelt, Mario (2023). Goods and bads of endocannabinoid system as a therapeutic target: Lessons learned after 30 years. Pharmacological reviews, 75(5), pp. 885-958. American Society for Pharmacology and Experimental Therapeutics 10.1124/pharmrev.122.000600

Krishnan, Sandhya R; Skiba, Adrianna; Luca, Simon Vlad; Marcourt, Laurence; Wolfender, Jean-Luc; Skalicka-Woźniak, Krystyna; Gertsch, Jürg (2023). Bioactivity-guided isolation of trypanocidal coumarins and dihydro-pyranochromones from selected Apiaceae plant species. Phytochemistry, 213, p. 113770. Elsevier 10.1016/j.phytochem.2023.113770

Gertsch, Jürg; Heilmann, Jörg; Skaltsa, Eleni (2023). Editorial. Phytochemistry, 213(113781), p. 113781. Elsevier 10.1016/j.phytochem.2023.113781

Fischer, Jérôme Paul; Bátora, Dániel; Dick, Luca Julian; Kaderli, Reto Martin; Gertsch, Jürg; Lochner, Martin (8 August 2023). Developing Molecular Tools for the Study and Detection of Calcium-Sensing Receptor [MC-112]. CHIMIA, 77(7/8), p. 526. Schweizerische Chemische Gesellschaft

Skiba, Adrianna; Pellegata, Daniele; Morozova, Veronika; Kozioł, Ewelina; Budzyńska, Barbara; Lee, Simon Ming-Yuen; Gertsch, Jürg; Skalicka-Woźniak, Krystyna (2023). Pharmacometabolic Effects of Pteryxin and Valproate on Pentylenetetrazole-Induced Seizures in Zebrafish Reveal Vagus Nerve Stimulation. Cells, 12(11) MDPI 10.3390/cells12111540

Reynoso-Moreno, Ines; Rau, Mark; Chicca, Andrea; Nicolussi, Simon; Gertsch, Jürg (2023). Assay of Endocannabinoid Uptake. Methods in molecular biology, 2576, pp. 329-348. Springer 10.1007/978-1-0716-2728-0_28

Jeckelmann, Jean-Marc; Zaugg, Jonas; Morozova, Veronika; Müller, Jennifer; Kantipudi, Satish; Schröder, Mariana; Graff, Julien; Albrecht, Christiane; Altmann, Karl-Heinz; Gertsch, Jürg; Fotiadis, Dimitrios (2022). Structure, Function and Pharmacology of SLC7 Family Members and Homologues. CHIMIA, 76(12), pp. 1011-1018. Schweizerische Chemische Gesellschaft 10.2533/chimia.2022.1011

Graff, Julien; Müller, Jennifer; Sadurní, Anna; Rubin, Matthias; Cuissa, Inês André Canivete; Keller, Claudia; Hartmann, Marco; Singer, Simon; Gertsch, Jürg; Altmann, Karl-Heinz (2022). The Evaluation of L-Tryptophan Derivatives as Inhibitors of the LType Amino Acid Transporter LAT1 (SLC7A5). ChemMedChem, 17(17), e202200308. Wiley-VCH 10.1002/cmdc.202200308

Fischer, Jérôme; Batora, Daniel; Kaderli, Reto Martin; Gertsch, Jürg; Lochner, Martin (July 2022). Developing Molecular Tools for the Study and Detection of Calcium-Sensing Receptor (CaSR) in Parathyroid Glands [MC-112]. CHIMIA, 76(7/8), p. 693. Schweizerische Chemische Gesellschaft

Bononi, Giulia; Di Stefano, Miriana; Poli, Giulio; Ortore, Gabriella; Meier, Philip; Masetto, Francesca; Caligiuri, Isabella; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Avan, Amir; Giovannetti, Elisa; Vagaggini, Chiara; Brai, Annalaura; Dreassi, Elena; Valoti, Massimo; Minutolo, Filippo; Granchi, Carlotta; Gertsch, Jürg and Tuccinardi, Tiziano (2022). Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives. Journal of medicinal chemistry, 65(10), pp. 7118-7140. American Chemical Society 10.1021/acs.jmedchem.1c01806

Gazzi, Thais; Brennecke, Benjamin; Atz, Kenneth; Korn, Claudia; Sykes, David; Forn-Cuni, Gabriel; Pfaff, Patrick; Sarott, Roman C; Westphal, Matthias V; Mostinski, Yelena; Mach, Leonard; Wasinska-Kalwa, Malgorzata; Weise, Marie; Hoare, Bradley L; Miljuš, Tamara; Mexi, Maira; Roth, Nicolas; Koers, Eline J; Guba, Wolfgang; Alker, André; ... (2022). Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe. Chemical Science, 13(19), pp. 5539-5545. The Royal Society of Chemistry 10.1039/d1sc06659e

Hinden, Liad; Ahmad, Majdoleen; Hamad, Sharleen; Nemirovski, Alina; Szanda, Gergő; Glasmacher, Sandra; Kogot-Levin, Aviram; Abramovitch, Rinat; Thorens, Bernard; Gertsch, Jürg; Leibowitz, Gil; Tam, Joseph (2022). Opposite physiological and pathological mTORC1-mediated roles of the CB1 receptor in regulating renal tubular function. Nature Communications, 13(1), p. 1783. Springer Nature 10.1038/s41467-022-29124-8

Kowalczyk, Joanna; Budzyńska, Barbara; Kurach, Łukasz; Pellegata, Daniele; El Sayed, Nesrine S; Gertsch, Jürg; Skalicka-Woźniak, Krystyna (2022). Neuropsychopharmacological profiling of scoparone in mice. Scientific reports, 12(1), p. 822. Springer Nature 10.1038/s41598-021-04741-3

Andrieu, Thomas; Chicca, Andrea; Pellegata, Daniele; Bersinger, Nick A.; Imboden, Sara; Nirgianakis, Konstantinos; Gertsch, Jürg; Mueller, Michael D. (2022). Association of endocannabinoids with pain in endometriosis. Pain, 163(1), pp. 193-203. Elsevier 10.1097/j.pain.0000000000002333

Luca, Simon Vlad; Gaweł-Bęben, Katarzyna; Strzępek-Gomółka, Marcelina; Czech, Karolina; Trifan, Adriana; Zengin, Gokhan; Korona-Glowniak, Izabela; Minceva, Mirjana; Gertsch, Jürg; Skalicka-Woźniak, Krystyna (2021). Insights into the Phytochemical and Multifunctional Biological Profile of Spices from the Genus Piper. Antioxidants, 10(10) MDPI 10.3390/antiox10101642

Alexander, Stephen Ph; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair; Peters, John A; Veale, Emma L; Armstrong, Jane F; Faccenda, Elena; Harding, Simon D; Pawson, Adam J; Southan, Christopher; Davies, Jamie A; Boison, Detlev; Burns, Kathryn Elisa; Dessauer, Carmen; Gertsch, Jürg; Helsby, Nuala Ann; Izzo, Angelo A; Koesling, Doris; Ostrom, Rennolds; ... (2021). THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Enzymes. British journal of pharmacology, 178(Suppl. 1), S313-S411. Wiley 10.1111/bph.15542

Schafroth, Michael A; Mazzoccanti, Giulia; Reynoso-Moreno, Ines; Erni, Reto; Pollastro, Federica; Caprioglio, Diego; Botta, Bruno; Allegrone, Gianna; Grassi, Giulio; Chicca, Andrea; Gasparrini, Francesco; Gertsch, Jürg; Carreira, Erick M; Appendino, Giovanni (2021). Δ9-cis-Tetrahydrocannabinol: Natural Occurrence, Chirality, and Pharmacology. Journal of natural products, 84(9), pp. 2502-2510. American Chemical Society 10.1021/acs.jnatprod.1c00513

Glasmacher, Sandra; Gertsch, Jürg (2021). Characterization of pepcan-23 as pro-peptide of RVD-hemopressin (pepcan-12) and stability of hemopressins in mice. Advances in biological regulation, 80, p. 100808. Elsevier 10.1016/j.jbior.2021.100808

Salm, Andrea; Krishnan, Sandhya R.; Collu, Marta; Danton, Ombeline; Hamburger, Matthias; Leonti, Marco; Almanza, Giovanna; Gertsch, Jürg (2021). Phylobioactive hotspots in plant resources used to treat Chagas disease. iScience, 24(4), p. 102310. Elsevier 10.1016/j.isci.2021.102310

Gruber, Thomas; Robatel, Steve; Kremenovic, Mirela; Bäriswyl, Lukas; Gertsch, Jürg; Schenk, Mirjam (2021). Cannabinoid Receptor Type-2 in B Cells Is Associated with Tumor Immunity in Melanoma. Cancers, 13(8) MDPI AG 10.3390/cancers13081934

Reynoso-Moreno, Ines; Tietz, Silvia; Vallini, Erika; Engelhardt, Britta; Gertsch, Jürg; Chicca, Andrea (2021). Selective Endocannabinoid Reuptake Inhibitor WOBE437 Reduces Disease Progression in a Mouse Model of Multiple Sclerosis. ACS pharmacology & translational science, 4(2), pp. 765-779. ACS Publications 10.1021/acsptsci.0c00214

Altmann, Karl-Heinz; Bold, Christian Paul; Gut, Melanie; Schürmann, Jasmine; Lucena Agell, Daniel; Diaz, Jose Fernando; Gertsch, Jürg (2021). Synthesis of Morpholine-Based Analogs of (-)-Zampanolide and Their Biological Activity. Chemistry: a European journal, 27(19), pp. 5936-5943. Wiley 10.1002/chem.202003996

Yan, Renhong; Li, Yaning; Müller, Jennifer; Zhang, Yuanyuan; Singer, Simon; Xia, Lu; Zhong, Xinyue; Gertsch, Jürg; Altmann, Karl-Heinz; Zhou, Qiang (2021). Mechanism of substrate transport and inhibition of the human LAT1-4F2hc amino acid transporter. Cell discovery, 7(1), p. 16. Springer Nature 10.1038/s41421-021-00247-4

Luca, Simon Vlad; Minceva, Mirjana; Gertsch, Jürg; Skalicka-Wozniak, Krystyna Katarzyna (2021). LC-HRMS/MS-based phytochemical profiling of Piper spices: Global association of piperamides with endocannabinoid system modulation. Food research international, 141, p. 110123. Elsevier 10.1016/j.foodres.2021.110123

Schuele, Lena-Louise; Glasmacher, Sandra; Gertsch, Jürg; Roggan, Marie Denise; Transfeld, Janis-Lisa; Bindila, Laura; Lutz, Beat; Kolbe, Carl-Christian; Bilkei-Gorzo, Andras; Zimmer, Andreas; Leidmaa, Este (2021). Diacylglycerol lipase alpha in astrocytes is involved in maternal care and affective behaviors. GLIA, 69(2), pp. 377-391. Wiley 10.1002/glia.23903

Mäder, Patrick; Bartholomäus, Ruben; Nicolussi, Simon; Baumann, Alice; Weis, Melanie; Chicca, Andrea; Rau, Mark; Simão, Ana Catarina; Gertsch, Jürg; Altmann, Karl-Heinz (2021). Synthesis and Biological Evaluation of Endocannabinoid Uptake Inhibitors Derived from WOBE437. ChemMedChem, 16(1), pp. 145-154. Wiley-VCH 10.1002/cmdc.202000153

Granchi, Carlotta; Bononi, Giulia; Ferrisi, Rebecca; Gori, Eleonora; Mantini, Giulia; Glasmacher, Sandra; Poli, Giulio; Palazzolo, Stefano; Caligiuri, Isabella; Rizzolio, Flavio; Canzonieri, Vincenzo; Perin, Tiziana; Gertsch, Jürg; Sodi, Andrea; Giovannetti, Elisa; Macchia, Marco; Minutolo, Filippo; Tuccinardi, Tiziano; Chicca, Andrea (2021). Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors. European journal of medicinal chemistry, 209, p. 112857. Elsevier 10.1016/j.ejmech.2020.112857

Arena, Chiara; Gado, Francesca; Di Cesare Mannelli, Lorenzo; Cervetto, Chiara; Carpi, Sara; Reynoso-Moreno, Ines; Polini, Beatrice; Vallini, Erika; Chicca, Stefano; Lucarini, Elena; Bertini, Simone; D'Andrea, Felicia; Digiacomo, Maria; Poli, Giulio; Tuccinardi, Tiziano; Macchia, Marco; Gertsch, Jürg; Marcoli, Manuela; Nieri, Paola; Ghelardini, Carla; ... (2020). The endocannabinoid system dual-target ligand N-cycloheptyl-1,2-dihydro-5-bromo-1-(4-fluorobenzyl)-6-methyl-2-oxo-pyridine-3-carboxamide improves disease severity in a mouse model of multiple sclerosis. European journal of medicinal chemistry, 208, p. 112858. Elsevier 10.1016/j.ejmech.2020.112858

Miller, Sally; Daily, Laura; Dharla, Vijai; Gertsch, Jürg; Malamas, Michael S; Ojima, Iwao; Kaczocha, Martin; Ogasawara, Daisuke; Straiker, Alex (2020). Endocannabinoid metabolism and transport as targets to regulate intraocular pressure. Experimental eye research, 201, p. 108266. Elsevier 10.1016/j.exer.2020.108266

Zaugg, Jonas; Huang, Xiao; Ziegler, Fabian; Rubin, Matthias; Graff, Julien; Müller, Jennifer; Moser-Hässig, Ruedi; Powell, Theresa; Gertsch, Jürg; Altmann, Karl-Heinz; Albrecht, Christiane (2020). Small molecule inhibitors provide insights into the relevance of LAT1 and LAT2 in materno-foetal amino acid transport. Journal of cellular and molecular medicine, 24(21), pp. 12681-12693. Wiley 10.1111/jcmm.15840

Sarott, Roman C; Westphal, Matthias V; Pfaff, Patrick; Korn, Claudia; Sykes, David A; Gazzi, Thais; Brennecke, Benjamin; Atz, Kenneth; Weise, Marie; Mostinski, Yelena; Hompluem, Pattarin; Koers, Eline; Miljuš, Tamara; Roth, Nicolas J; Asmelash, Hermon; Vong, Man C; Piovesan, Jacopo; Guba, Wolfgang; Rufer, Arne C; Kusznir, Eric A; ... (2020). Development of High-Specificity Fluorescent Probes to Enable Cannabinoid Type 2 Receptor Studies in Living Cells. Journal of the American Chemical Society, 142(40), pp. 16953-16964. American Chemical Society 10.1021/jacs.0c05587

Guha, Sujay; Calarco, Serafina; Gachet, M. Salomé; Gertsch, Jürg (2020). Juniperonic Acid Biosynthesis is Essential in Caenorhabditis Elegans Lacking Δ6 Desaturase (fat-3) and Generates New ω-3 Endocannabinoids. Cells, 9(9) MDPI 10.3390/cells9092127

Skalicka-Wozniak, Krystyna; Gertsch, Jürg (2020). Antipsychotic natural products. In: Annual Reports in Medicinal Chemistry 55 (pp. 481-515). Elsevier 10.1016/bs.armc.2020.03.004

Petrelli, Francesco; Dallérac, Glenn; Pucci, Luca; Calì, Corrado; Zehnder, Tamara; Sultan, Sébastien; Lecca, Salvatore; Chicca, Andrea; Ivanov, Andrei; Asensio, Cédric S; Gundersen, Vidar; Toni, Nicolas; Knott, Graham William; Magara, Fulvio; Gertsch, Jürg; Kirchhoff, Frank; Déglon, Nicole; Giros, Bruno; Edwards, Robert H; Mothet, Jean-Pierre; ... (2020). Dysfunction of homeostatic control of dopamine by astrocytes in the developing prefrontal cortex leads to cognitive impairments. Molecular psychiatry, 25(4), pp. 732-749. Nature Publishing Group 10.1038/s41380-018-0226-y

Saliakoura, Maria; Reynoso-Moreno, Inés; Pozzato, Chiara; Rossi Sebastiano, Matteo; Galié, Mirco; Gertsch, Jürg; Konstantinidou, Georgia (2020). The ACSL3-LPIAT1 signaling drives prostaglandin synthesis in non-small cell lung cancer. Oncogene, 39(14), pp. 2948-2960. Springer Nature 10.1038/s41388-020-1196-5

Gado, Francesca; Arena, Chiara; Fauci, Cristiana La; Reynoso-Moreno, Ines; Bertini, Simone; Digiacomo, Maria; Meini, Serena; Poli, Giulio; Macchia, Marco; Tuccinardi, Tiziano; Gertsch, Jürg; Chicca, Andrea; Manera, Clementina (2020). Modification on the 1,2-dihydro-2-oxo-pyridine-3-carboxamide core to obtain multi-target modulators of endocannabinoid system. Bioorganic chemistry, 94, p. 103353. Elsevier 10.1016/j.bioorg.2019.103353

Bartholomäus, Ruben; Nicolussi, Simon; Baumann, Alice; Rau, Mark; Simão, Ana Catarina; Gertsch, Jürg; Altmann, Karl-Heinz (2019). Total Synthesis of the Endocannabinoid Uptake Inhibitor Guineensine and SAR Studies. ChemMedChem, 14(17), pp. 1590-1596. Wiley-VCH 10.1002/cmdc.201900390

Salm, Andrea; Gertsch, Jürg (2019). Cultural perception of triatomine bugs and Chagas disease in Bolivia: a cross-sectional field study. Parasites & Vectors, 12(1), p. 291. BioMed Central 10.1186/s13071-019-3546-0

Marino, Silvia; de Ridder, Daniëlle; Bishop, Ryan T; Renema, Nathalie; Ponzetti, Marco; Sophocleous, Antonia; Capulli, Mattia; Aljeffery, Abdullah; Carrasco, Giovana; Dalghi Gens, Marianela; Khogeer, Asim; Ralston, Stuart H; Gertsch, Jürg; Lamoureux, Francois; Heymann, Dominique; Rucci, Nadia; Idris, Aymen I (2019). Paradoxical effects of JZL184, an inhibitor of monoacylglycerol lipase, on bone remodelling in healthy and cancer-bearing mice. EBioMedicine, 44, pp. 452-466. Elsevier 10.1016/j.ebiom.2019.05.048

Gertsch, Jürg (2019). Scaffold and organism hopping with chemical probes. Nature chemical biology, 15(5), pp. 428-429. Springer Nature 10.1038/s41589-019-0275-9

Dornbierer, Dario A; Kometer, Michael; Von Rotz, Robin; Studerus, Erich; Gertsch, Jürg; Gachet Otanez, M. Salomé; Vollenweider, Franz X; Seifritz, Erich; Bosch, Oliver G; Quednow, Boris B (2019). Effects of gamma-hydroxybutyrate on neurophysiological correlates of performance and conflict monitoring. European neuropsychopharmacology, 29(4), pp. 539-548. Elsevier 10.1016/j.euroneuro.2019.02.004

Delalande, Clémence; Awale, Mahendra; Rubin, Matthias; Probst, Daniel; Ozhathil, Lijo C.; Gertsch, Jürg; Abriel, Hugues; Reymond, Jean-Louis (2019). Optimizing TRPM4 inhibitors in the MHFP6 chemical space. European journal of medicinal chemistry, 166, pp. 167-177. Elsevier 10.1016/j.ejmech.2019.01.048

Granchi, Carlotta; Lapillo, Margherita; Glasmacher, Sandra; Bononi, Giulia; Licari, Cristina; Poli, Giulio; El Boustani, Maguie; Caligiuri, Isabella; Rizzolio, Flavio; Gertsch, Jürg; Macchia, Marco; Minutolo, Filippo; Tuccinardi, Tiziano; Chicca, Andrea (2019). Optimization of a Benzoylpiperidine Class Identifies a Highly Potent and Selective Reversible Monoacylglycerol Lipase (MAGL) Inhibitor. Journal of medicinal chemistry, 62(4), pp. 1932-1958. American Chemical Society 10.1021/acs.jmedchem.8b01483

Grafinger, Katharina Elisabeth; Mandhair, Harpreet Kaur; Broillet, Alain; Gertsch, Jürg; Weinmann, Wolfgang (2019). Cytotoxicity of the synthetic cannabinoids 5C-AKB48, 5F-MDMB-PINACA, ADB-CHMINACA, MDMB-CHMICA and NM-2201 in A549 and TR146 cell lines. Forensic toxicology, 37(2), pp. 398-411. Springer 10.1007/s11419-019-00474-1

Chicca, Andrea; Schafroth, M A; Reynoso, Ines del Carmen; Erni, R; Petrucci, Vanessa; Carreira, E M; Gertsch, Jürg (2018). Uncovering the psychoactivity of a cannabinoid from liverworts associated with a legal high. Science Advances, 4(10), eaat2166. American Association for the Advancement of Science 10.1126/sciadv.aat2166

Zákány, Nóra; Oláh, Attila; Markovics, Arnold; Takács, Erika; Aranyász, Andrea; Nicolussi, Simon; Piscitelli, Fabiana; Allarà, Marco; Pór, Ágnes; Kovács, Ilona; Zouboulis, Christos C; Gertsch, Jürg; Di Marzo, Vincenzo; Bíró, Tamás; Szabó, Tamás (2018). Endocannabinoid Tone Regulates Human Sebocyte Biology. Journal of Investigative Dermatology, 138(8), pp. 1699-1706. Nature Publishing 10.1016/j.jid.2018.02.022

Chicca, Andrea; Arena, Chiara; Bertini, Simone; Gado, Francesca; Ciaglia, Elena; Abate, Mario; Digiacomo, Maria; Lapillo, Margherita; Poli, Giulio; Bifulco, Maurizio; Macchia, Marco; Tuccinardi, Tiziano; Gertsch, Jürg; Manera, Clementina (2018). Polypharmacological profile of 1,2-dihydro-2-oxo-pyridine-3-carboxamides in the endocannabinoid system. European journal of medicinal chemistry, 154, pp. 155-171. Elsevier 10.1016/j.ejmech.2018.05.019

Ozhathil, Lijo Cherian; Delalande, Clémence Marie Sandrine; Bianchi, Beatrice; Nemeth, Gabor; Kappel, Sven; Thomet, Urs; Ross, Daniela; Simonin, Céline; Rubin, Matthias; Gertsch, Jürg; Lochner, Martin; Peinelt, Christine; Reymond, Jean-Louis; Abriel, Hugues (2018). Identification of potent and selective small molecule inhibitors of the cation channel TRPM4. British journal of pharmacology, 175(12), pp. 2504-2519. Wiley-Blackwell 10.1111/bph.14220

Benabdelaziz, Imane; Gómez-Ruiz, Santiago; Benkhaled, Mohammed; Carralero, Sandra; Schenker, Patricia; Salm, Andrea Alejandra; Gertsch, Jürg; Haba, Hamada (2018). New cycloartane-type ester triterpenes from Euphorbia pterococca and biological evaluation. Fitoterapia, 127, pp. 271-278. Elsevier Science 10.1016/j.fitote.2018.02.027

Aghazadeh Tabrizi, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Ruggiero, Emanuela; De Stefano, Lucia; Rizzolio, Flavio; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Chicca, Andrea; Lapillo, Margherita; Gertsch, Jürg; Manera, Clementina; Macchia, Marco; Martinelli, Adriano; Granchi, Carlotta; Minutolo, Filippo; Tuccinardi, Tiziano (2018). Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors. Journal of medicinal chemistry, 61(3), pp. 1340-1354. American Chemical Society 10.1021/acs.jmedchem.7b01845

Varga, Zoltan V; Matyas, Csaba; Erdelyi, Katalin; Cinar, Resat; Nieri, Daniela; Chicca, Andrea; Nemeth, Balazs Tamas; Paloczi, Janos; Lajtos, Tamas; Corey, Lukas; Hasko, Gyorgy; Gao, Bin; Kunos, George; Gertsch, Jürg; Pacher, Pal (2018). Beta-caryophyllene protects against alcoholic steatohepatitis by attenuating inflammation and metabolic dysregulation in mice. British journal of pharmacology, 175(2), pp. 320-334. Wiley-Blackwell 10.1111/bph.13722

Reynoso, Ines del Carmen; Chicca, Andrea; Flores-Soto, Mario E; Viveros-Paredes, Juan M; Gertsch, Jürg (2018). The Endocannabinoid Reuptake Inhibitor WOBE437 Is Orally Bioavailable and Exerts Indirect Polypharmacological Effects via Different Endocannabinoid Receptors. Frontiers in molecular neuroscience, 11, p. 180. Frontiers Research Foundation 10.3389/fnmol.2018.00180

Bertini, Simone; Chicca, Andrea; Gado, Francesca; Arena, Chiara; Nieri, Daniela; Digiacomo, Maria; Saccomanni, Giuseppe; Zhao, Pingwei; Abood, Mary E; Macchia, Marco; Gertsch, Jürg; Manera, Clementina (2017). Novel analogs of PSNCBAM-1 as allosteric modulators of cannabinoid CB1 receptor. Bioorganic & medicinal chemistry, 25(24), pp. 6427-6434. Elsevier 10.1016/j.bmc.2017.10.015

Chicca, Andrea; Berg, Regina; Jessen, Henning J; Marck, Nicolas; Schmid, Fabian; Burch, Patrick; Gertsch, Jürg; Gademann, Karl (2017). Biological evaluation of pyridone alkaloids on the endocannabinoid system. Bioorganic & medicinal chemistry, 25(22), pp. 6102-6114. Elsevier 10.1016/j.bmc.2017.02.031

Reynoso, Ines del Carmen; Najar-Guerrero, Israel; Escareño, Noé; Flores-Soto, Mario Eduardo; Gertsch, Jürg; Viveros-Paredes, Juan Manuel (2017). An Endocannabinoid Uptake Inhibitor from Black Pepper Exerts Pronounced Anti-Inflammatory Effects in Mice. Journal of agricultural and food chemistry, 65(43), pp. 9435-9442. American Chemical Society 10.1021/acs.jafc.7b02979

Patsenker, Eleonora; Chicca, Andrea; Petrucci, Vanessa; Moghadamrad, Sheida; De Gottardi, Andrea; Hampe, Jochen; Gertsch, Jürg; Semmo, Nasser; Stickel, Felix (2017). 4-O'-methylhonokiol protects from alcohol/carbon tetrachloride-induced liver injury in mice. Journal of molecular medicine JMM, 95(10), pp. 1077-1089. Springer 10.1007/s00109-017-1556-y

Petrucci, Vanessa; Chicca, Andrea; Glasmacher, Sandra Patricia; Paloczi, Janos; Cao, Zongxian; Pacher, Pal; Gertsch, Jürg (2017). Pepcan-12 (RVD-hemopressin) is a CB2 receptor positive allosteric modulator constitutively secreted by adrenals and in liver upon tissue damage. Scientific Reports, 7(1), p. 9560. Nature Publishing Group 10.1038/s41598-017-09808-8

von Rotz, Robin; Kometer, Michael; Dornbierer, Dario; Gertsch, Jürg; Gachet Otanez, Maria Salomé; Vollenweider, Franz X; Seifritz, Erich; Bosch, Oliver G; Quednow, Boris B (2017). Neuronal oscillations and synchronicity associated with gamma-hydroxybutyrate during resting-state in healthy male volunteers. Psychopharmacology, 234(13), pp. 1957-1968. Springer 10.1007/s00213-017-4603-z

Chicca, Andrea; Nicolussi, Simon; Bartholomäus, Ruben; Blunder, Martina; Aparisi Rey, Alejandro; Petrucci, Vanessa; Reynoso, Ines del Carmen; Viveros-Paredes, Juan Manuel; Dalghi Gens, Marianela Gisela; Lutz, Beat; Schiöth, Helgi B; Soeberdt, Michael; Abels, Christoph; Charles, Roch-Philippe; Altmann, Karl-Heinz; Gertsch, Jürg (2017). Chemical probes to potently and selectively inhibit endocannabinoid cellular reuptake. Proceedings of the National Academy of Sciences of the United States of America - PNAS, 114(25), E5006-E5015. National Academy of Sciences NAS 10.1073/pnas.1704065114

Gertsch, Jürg (2017). Cannabimimetic phytochemicals in the diet - an evolutionary link to food selection and metabolic stress adaptation? British journal of pharmacology, 174(11), pp. 1464-1483. Wiley-Blackwell 10.1111/bph.13676

El Mokh, Oussama; Ruffieux-Daidié, Dorothée; Rölli, Matthias Andreas; Stooss, Amandine; Phillips, Wayne A; Gertsch, Jürg; Dettmer, Matthias; Charles, Roch-Philippe (2017). Combined MEK and Pi3'-kinase inhibition reveals synergy in targeting thyroid cancer in vitro and in vivo. OncoTarget, 8(15), pp. 24604-24620. Impact Journals LLC 10.18632/oncotarget.15599

Gachet Otanez, Maria Salomé; Schubert, Alexandra; Calarco, Serafina; Boccard, Julien; Gertsch, Jürg (2017). Targeted metabolomics shows plasticity in the evolution of signaling lipids and uncovers old and new endocannabinoids in the plant kingdom. Scientific Reports, 7, p. 41177. Nature Publishing Group 10.1038/srep41177

Soethoudt, Marjolein; Grether, Uwe; Fingerle, Jürgen; Grim, Travis W; Fezza, Filomena; de Petrocellis, Luciano; Ullmer, Christoph; Rothenhäusler, Benno; Perret, Camille; van Gils, Noortje; Finlay, David; MacDonald, Christa; Chicca, Andrea; Gens, Marianela Dalghi; Stuart, Jordyn; de Vries, Henk; Mastrangelo, Nicolina; Xia, Lizi; Alachouzos, Georgios; Baggelaar, Marc P; ... (2017). Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity. Nature communications, 8(13958), p. 13958. Nature Publishing Group 10.1038/ncomms13958

Martínez-Pacheco, Heidy; Ramírez-Galicia, Guillermo; Vergara-Arias, Midalia; Gertsch, Jürg; Fragoso-Vázquez, Jonathan Manuel; Méndez-Luna, David; Abujamra, A L; Cristina, Cabrera-Pérez Laura; Cecilia, Rosales-Hernández Martha; Mendoza-Lujambio, I; Correa-Basurto, José (2017). Docking and QSAR studies of aryl-valproic acid derivatives to identify anti-proliferative agents targeting the HDAC8. Anti-cancer agents in medicinal chemistry, 17(7), pp. 927-940. Bentham Science Publishers

Alferink, Judith; Specht, Sabine; Arends, Hannah; Schumak, Beatrix; Schmidt, Kim; Ruland, Christina; Lundt, Ramona; Kemter, Andrea; Dlugos, Andrea; Kuepper, Janina M; Poppensieker, Karola; Findeiss, Matthias; Albayram, Önder; Otte, David-M; Marazzi, Janine; Gertsch, Jürg; Förster, Irmgard; Maier, Wolfgang; Scheu, Stefanie; Hoerauf, Achim; ... (2016). Cannabinoid Receptor 2 Modulates Susceptibility to Experimental Cerebral Malaria through a CCL17-dependent Mechanism. Journal of biological chemistry, 291(37), pp. 19517-19531. American Society for Biochemistry and Molecular Biology 10.1074/jbc.M116.746594

Jantsch, Andrea; Nieto, Lidia; Gertsch, Jürg; Rodríguez-Salarichs, Javier; Matesanz, Ruth; Jiménez-Barbero, Jesús; Díaz, J Fernando; Canales, Ángeles; Altmann, Karl-Heinz (2016). Synthesis, Biological Profiling and Determination of the Tubulin-Bound Conformation of 12-Aza-Epothilones (Azathilones). Molecules, 21(8) MDPI 10.3390/molecules21081010

Gertsch, Jürg (2016). The Metabolic Plant Feedback Hypothesis: How Plant Secondary Metabolites Nonspecifically Impact Human Health. Planta medica, 82(11-12), pp. 920-929. Thieme 10.1055/s-0042-108340

Bertini, Simone; Chicca, Andrea; Arena, Chiara; Chicca, Stefano; Saccomanni, Giuseppe; Gertsch, Jürg; Manera, Clementina; Macchia, Marco (2016). Synthesis and pharmacological evaluation of new biphenylic derivatives as CB2 receptor ligands. European journal of medicinal chemistry, 116, pp. 252-266. Elsevier Masson SAS 10.1016/j.ejmech.2016.03.072

Oláh, Attila; Ambrus, Lídia; Nicolussi, Simon; Gertsch, Jürg; Tubak, Vilmos; Kemény, Lajos; Soeberdt, Michael; Abels, Christoph; Bíró, Tamás (2016). Inhibition of fatty acid amide hydrolase exerts cutaneous anti-inflammatory effects both in vitro and in vivo. Experimental dermatology, 25(4), pp. 328-330. Blackwell 10.1111/exd.12930

Gertsch, Jürg (2016). Editorial: Lung macrophages high on cannabinoids: jamming PAMs and taming TAMs? Journal of leukocyte biology, 99(4), pp. 518-520. Society for Leukocyte Biology 10.1189/jlb.3CE0915-409RR

Rau, Mark; Nicolussi, Simon; Chicca, Andrea; Gertsch, Jürg (2016). Assay of Endocannabinoid Uptake. In: Maccarrone, Mauro (ed.) Endocannabinoid Signaling. Methods and Protocols. Methods in Molecular Biology: Vol. 1412 (pp. 191-203). New York: Springer 10.1007/978-1-4939-3539-0_20

Liechti, Matthias E; Quednow, Boris B; Liakoni, Evangelia; Dornbierer, Dario; von Rotz, Robin; Gachet Otanez, Maria Salomé; Gertsch, Jürg; Seifritz, Erich; Bosch, Oliver G (2015). Pharmacokinetics and pharmacodynamics of γ-hydroxybutyrate in healthy subjects. British journal of clinical pharmacology, 81(5), pp. 980-988. Wiley-Blackwell 10.1111/bcp.12863

Bosch, Oliver G; Eisenegger, Christoph; Gertsch, Jürg; von Rotz, Robin; Dornbierer, Dario; Gachet Otanez, Maria Salomé; Heinrichs, Markus; Wetter, Thomas C; Seifritz, Erich; Quednow, Boris B (2015). Gamma-hydroxybutyrate enhances mood and prosocial behavior without affecting plasma oxytocin and testosterone. Psychoneuroendocrinology, 62, pp. 1-10. Elsevier 10.1016/j.psyneuen.2015.07.167

Gachet Otanez, Maria Salomé; Gertsch, Jürg (2015). Quantitative analysis of arachidonic acid, endocannabinoids, N-acylethanolamines and steroids in biological samples by LCMS/MS: Fit to purpose. Journal of chromatography. B - analytical technologies in the biomedical and life sciences, 1012-1013, pp. 215-221. Elsevier 10.1016/j.jchromb.2015.11.013

Iakovenko, Roman O; Kazakova, Anna N; Muzalevskiy, Vasiliy M; Ivanov, Alexander Yu; Boyarskaya, Irina A; Chicca, Andrea; Petrucci, Vanessa; Gertsch, Jürg; Krasavin, Mikhail; Starova, Galina L; Zolotarev, Andrey A; Avdontceva, Margarita S; Nenajdenko, Valentine G; Vasilyev, Aleksander V (2015). Reactions of CF3-enones with arenes under superelectrophilic activation: a pathway to trans-1,3-diaryl-1-CF3-indanes, new cannabinoid receptor ligands. Organic & biomolecular chemistry, 13(33), pp. 8827-8842. Royal Society of Chemistry 10.1039/c5ob01072a

Del Carlo, S; Manera, C; Chicca, Andrea; Arena, C; Bertini, S; Burgalassi, S; Tampucci, S; Gertsch, Jürg; Macchia, M; Saccomanni, G (2015). Development of an HPLC/UV assay for the evaluation of inhibitors of human recombinant monoacylglycerol lipase. Journal of pharmaceutical and biomedical analysis, 108, pp. 113-121. Pergamon Press 10.1016/j.jpba.2015.02.007

Hofer Reyes, Stefanie; Ralvenius, William T; Gachet Otanez, Maria Salomé; Fritschy, Jean-Marc; Zeilhofer, Ulrich; Gertsch, Jürg (2015). Localization and production of peptide endocannabinoids in the rodent CNS and adrenal medulla. Neuropharmacology, 98, pp. 78-89. Elsevier 10.1016/j.neuropharm.2015.03.021

Jack, Thomas; Simonin, Jonathan; Ruepp, Marc-David; Thompson, Andrew James; Gertsch, Jürg; Lochner, Martin (2015). Characterizing New Fluorescent Tools for Studying 5-HT3 Receptor Pharmacology. Neuropharmacology, 90, pp. 63-73. Elsevier 10.1016/j.neuropharm.2014.11.007

Gachet Otanez, Maria Salomé; Rhyn, Peter; Bosch, Oliver G; Quednow, Boris B; Gertsch, Jürg (2015). A quantitiative LC-MS/MS method for the measurement of arachidonic acid, prostanoids, endocannabinoids, N-acylethanolamines and steroids in human plasma. Journal of chromatography. B - analytical technologies in the biomedical and life sciences, 976-977, pp. 6-18. Elsevier 10.1016/j.jchromb.2014.11.001

Nicolussi, Simon; Gertsch, Jürg (2015). Endocannabinoid transport revisited. In: Litwack, Gerald (ed.) Vitamins and Hormones. Hormones and Transport Systems: Vol. 98 (pp. 441-485). Elsevier Inc. 10.1016/bs.vh.2014.12.011

Patsenker, Eleanora; Sachse, Philip; Chicca, Andrea; Gachet Otanez, Maria Salomé; Schneider, Vreni; Mattsson, Johan; Lanz, Christian; Worni, Mathias; De Gottardi, Andrea; Semmo, Mariam; Hampe, Jochen; Schafmayer, Clemens; Brenneisen, Rudolf Max; Gertsch, Jürg; Stickel, Felix; Semmo, Nasser (2015). Elevated levels of endocannabinoids in chronic hepatitis C may modulate cellular immune response and hepatic stellate cell activation. International journal of molecular sciences, 16(4), pp. 7057-7076. MDPI 10.3390/ijms16047057

Chicca, Andrea; Gachet Otanez, Maria Salomé; Petrucci, Vanessa; Schuehly, Wolfgang; Charles, Roch-Philippe; Gertsch, Jürg (2015). 4'-O-methylhonokiol increases levels of 2-arachidonoyl glycerol in mouse brain via selective inhibition of its COX-2-mediated oxygenation. Journal of neuroinflammation, 12, p. 89. BioMed Central 10.1186/s12974-015-0307-7

Nicolussi, Simon; Chicca, Andrea; Rau, Mark; Rihs, Sabine; Soeberdt, Michael; Abels, Christoph; Gertsch, Jürg (2014). Correlating FAAH and anandamide cellular uptake inhibition using N-alkylcarbamate inhibitors: from ultrapotent to hyperpotent. Biochemical pharmacology, 92(4), pp. 669-689. Elsevier 10.1016/j.bcp.2014.09.020

Rosati, Ornelio; Messina, Federica; Pelosi, Azzurra; Curini, Massimo; Petrucci, Vanessa; Gertsch, Jürg; Chicca, Andrea (2014). One-pot heterogeneous synthesis of Δ(3)-tetrahydrocannabinol analogues and xanthenes showing differential binding to CB(1) and CB(2) receptors. European journal of medicinal chemistry, 85, pp. 77-86. Elsevier Masson SAS 10.1016/j.ejmech.2014.07.062

Marini, Camilla; Lüscher, Benjamin; Jörger Messerli, Marianne; Sager, Ruth; Huang, Xiao; Gertsch, Jürg; Hediger, Matthias; Albrecht, Christiane; Baumann, Marc Ulrich; Surbek, Daniel (September 2014). PLACENTAL GLUCOSE TRANSPORTER (GLUT)-1 REGULATION IN PREECLAMPSIA. Placenta, 35, A83-A84. Elsevier

Hajdu, Zsanett; Nicolussi, Simon; Rau, Mark; Lorántfy, László; Forgo, Peter; Hohmann, Judit; Csupor, Dezső; Gertsch, Jürg (2014). Identification of endocannabinoid system-modulating N-alkylamides from Heliopsis helianthoides var. scabra and Lepidium meyenii. Journal of natural products, 77(7), pp. 1663-1669. American Chemical Society 10.1021/np500292g

Chicca, Andrea; Caprioglio, Diego; Minassi, Alberto; Petrucci, Vanessa; Appendino, Giovanni; Taglialatela-Scafati, Orazio; Gertsch, Jürg (2014). Functionalization of β-caryophyllene generates novel polypharmacology in the endocannabinoid system. ACS Chemical Biology, 9(7), pp. 1499-1507. American Chemical Society 10.1021/cb500177c

Bürgi, Justus; Awale, Mahendra; Boss, Silvan D.; Schaer, Tifany; Marger, Fabrice; Viveros Paredes, Juan Manuel; Bertrand, Sonia; Gertsch, Jürg; Bertrand, Daniel; Reymond, Jean-Louis (2014). Discovery of Potent Positive Allosteric Modulators of the α3β2 Nicotinic Acetylcholine Receptor by a Chemical Space Walk in ChEMBL. ACS chemical neuroscience, 5(5), pp. 346-359. American Chemical Society 10.1021/cn4002297

Ilgü, Hüseyin; Jeckelmann, Jean-Marc; Gachet Otanez, Maria Salomé; Boggavarapu, Venkata Ravi Naga Rajendr; Ucurum Fotiadis, Zöhre; Gertsch, Jürg; Fotiadis, Dimitrios José (2014). Variation of the detergent-binding capacity and phospholipid content of membrane proteins when purified in different detergents. Biophysical journal, 106(8), pp. 1660-1670. Biophysical Society 10.1016/j.bpj.2014.02.024

Klauke, A.-L.; Racz, I.; Pradier, B.; Markert, A.; Zimmer, A. M.; Gertsch, J.; Zimmer, A. (2014). The cannabinoid CB2 receptor-selective phytocannabinoid beta-caryophyllene exerts analgesic effects in mouse models of inflammatory and neuropathic pain. European neuropsychopharmacology, 24(4), pp. 608-620. Elsevier 10.1016/j.euroneuro.2013.10.008

Marini, Camilla; Lüscher, Benjamin; Jörger Messerli, Marianne; Sager, Ruth; Huang, Xiao; Gertsch, Jürg; Hediger, Matthias; Albrecht, Christiane; Baumann, Marc Ulrich; Surbek, Daniel (March 2014). Placental Glucose Transporter (GLUT1) Expression in Pre-Eclampsia. Reproductive sciences, 21(3), 304A-304A. Sage

Burch, Patrick; Chicca, Andrea; Gertsch, Jürg; Gademann, Karl (2014). Functionally Optimized Neuritogenic Farinosone C Analogs: SAR-Study and Investigations on Their Mode of Action. ACS medicinal chemistry letters, 5(2), pp. 172-177. American Chemical Society 10.1021/ml400435h

Nicolussi, Simon; Viveros Paredes, Juan Manuel; Gachet Otanez, Maria Salomé; Rau, Mark; Flores-Soto, Mario Eduardo; Blunder, Martina; Gertsch, Jürg (2014). Guineensine is a novel inhibitor of endocannabinoid uptake showing cannabimimetic behavioral effects in BALB/c mice. Pharmacological research, 80, pp. 52-65. Elsevier 10.1016/j.phrs.2013.12.010

Wullschleger, Christoph W.; Gertsch, Jürg; Altmann, Karl-Heinz (2013). Synthesis and Biological Activity of 7,8,9-Trideoxy- and 7 R DesTHP-Peloruside A. Chemistry - a European journal, 19(39), pp. 13105-13111. Wiley-VCH 10.1002/chem.201301796

Baur, Roland; Gertsch, Jürg; Sigel, Erwin (2013). Do N-arachidonyl-glycine (NA-glycine) and 2-arachidonoyl glycerol (2-AG) share mode of action and the binding site on the β 2 subunit of GABA A receptors? PeerJ, 1, e149. PeerJ, Ltd 10.7717/peerj.149

Simonin, Jonathan; Jack, Thomas; Ruepp, Marc-David; Hothersall, Daniel; Connolly, Christopher; Chicca, Andrea; Gertsch, Jürg; Thompson, Andrew James; Lummis, Sarah C. R.; Lochner, Martin (August 2013). Synthesis of fluorescent probes for the study of the 5-HT3 receptor: applications in imaging and fluorescence polarization. CHIMIA, 67(7/8), p. 524. Schweizerische Chemische Gesellschaft

Leonti, Marco; Cabras, Stefano; Eugenia Castellanos, Maria; Challenger, Antony; Gertsch, Jürg; Casu, Laura (2013). Bioprospecting: Evolutionary implications from a post-olmec pharmacopoeia and the relevance of widespread taxa. Journal of ethnopharmacology, 147(1), pp. 92-107. Elsevier Science Ireland 10.1016/j.jep.2013.02.012

Pfeiffer, Bernhard; Speck-Gisler, Sandra; Barandun, Luzi; Senft, Ursula; de Groot, Claire; Lehmann, Irène; Ganci, Walter; Gertsch, Jürg; Altmann, Karl-Heinz (2013). Total Synthesis and Configurational Assignment of the Marine Natural Product Haliclamide. The Journal of organic chemistry, 78(6), pp. 2553-2563. American Chemical Society 10.1021/jo3027643

Gertsch, Jürg; Viveros Paredes, Juan Manuel; Taylor, Peter (2011). Plant immunostimulants-Scientific paradigm or myth? Journal of ethnopharmacology, 136(3), pp. 385-391. Shannon: Elsevier Science Ireland 10.1016/j.jep.2010.06.044

Erdélyi, Máté; Navarro-Vázquez, Armando; Pfeiffer, Bernhard; Kuzniewski, Christian N; Felser, Andrea; Widmer, Toni; Gertsch, Jürg; Pera, Benet; Díaz, José Fernando; Altmann, Karl-Heinz; Carlomagno, Teresa (2010). The binding mode of side chain- and C3-modified epothilones to tubulin. ChemMedChem, 5(6), pp. 911-920. Weinheim: Wiley-VCH 10.1002/cmdc.201000050

Leonti, Marco; Casu, Laura; Gertsch, Jürg; Bonsignore, Leonardo; Floris, Costantino; Casu, Mariano; Cottiglia, Filippo (2010). A pterocarpan from the seeds of Bituminaria morisiana. Journal of natural medicines, 64(3), pp. 354-7. Tōkyō: Springer 10.1007/s11418-010-0408-7

Shwe, Htay Htay; Aye, Mye; Sein, Myint Myint; Htay, Khin Than; Kreitmeier, Peter; Gertsch, Jürg; Reiser, Oliver; Heilmann, Jörg (2010). Cytotoxic steroidal saponins from the rhizomes of Tacca integrifolia. Chemistry & Biodiversity, 7(3), pp. 610-22. Zürich: Verlag Helvetica Chimica Acta